产品名称 C646, p300/CBP Inhibitor from LIFESPAN BIOSCIENCES INC.
产品货号 LS-H2613
产品价格 现货询价,电话:010-67529703
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产品品牌 LIFESPAN BIOSCIENCES INC.
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Product NameC646, p300/CBP Inhibitor
DescriptionPurity >98% by NMR. Cell-permeable. A reversible, p300/CBP (CREB-binding protein) histone acetyltransferase (HAT) inhibitor (Ki = 400 nM). Specific inhibition to p300 (86%) compared to N-acetyltransferase, PCAF, GCN5, Rtt109, Sas or MOZ histone acetyltransferases (<10%). Suppresses histone H3 and H4 acetylation in mouse fibroblast cell lines.
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Other Names(E)-4-(4-((5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl)-methylene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid
Gene, Accession, CAS #CAS: 328968-36-1
Catalog #LS-H2613
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Order / More InfoC646, p300/CBP Inhibitor from LIFESPAN BIOSCIENCES INC.
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